Share this post on:

product name Procainamide HCl


Description: Procainamide HCl is a sodium channel blocker, and also a DNA methyltransferase inhibitor, used in the treatment of cardiac arrhythmias. Procainamide hydrochloride is the hydrochloride salt preparation of Procainamide, a potent blocker of Na+ channels. Procainamide demonstrates antiarrhythmic effects correlated with blockade of the Na+ channels. Procainamide hydrochloride is an inhibitor of DNA methyltransferase. 

References: JPharmacol Rep. 2016 Jun;68(3):654-61.



Molecular Weight (MW)

271.79
Formula

C13H22ClN3O
CAS No.

614-39-1
Storage

-20℃ for 3 years in powder form
-80℃ for 2 years in solvent
Solubility (In vitro)

DMSO: 54 mg/mL (198.6 mM)
Water:
Ethanol: 54 mg/mL (198.6 mM)
Solubility (In vivo)

 
Synonyms

 

other peoduct :References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/1941100

In Vitro

In vitro activity:


Kinase Assay:


Cell Assay:

In Vivo  
Animal model  
Formulation & Dosage  
References  

Relebactam

Share this post on:

Author: Sodium channel