product name Mizolastine
Description: Mizolastine (also known as SL 850324) is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. Mizolastine (brand name: Mizollen) is a once-daily, non-sedating antihistamine. It blocks H1 receptors and is commonly fast-acting. It does not prevent the actual release of histamine from mast cells, just prevents it binding to receptors. Side effects can include dry mouth and throat.
References: BioDrugs. 1998 Jul;10(1):41-63.; Wikipedia
432.49
Formula
C24H25FN6O
CAS No.
108612-45-9
Storage
-20℃ for 3 years in powder form
-80℃ for 2 years in solvent
Solubility (In vitro)
DMSO: <1 mg/mL
Water: <1 mg/mL
Ethanol: <1 mg/mL
Solubility (In vivo)
Synonyms
SL 850324
other peoduct :References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/19427620
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