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product name Methscopolamine


Description: Methscopolamine is a muscarinic acetylcholine receptor blocker. Methscopolamine, a methylated derivative of scopolamine, is a muscarinic antagonist structurally similar to the neurotransmitter acetylcholine. Its mechanism of action involves blocking the muscarinic acetylcholine receptors. Methscopolamine is also commonly used as a drying agent, to dry up post-nasal drip, in cold, irritable bowel syndrome and allergy medications.

References: J Pharm Pharmacol. 1964 Oct;16:690-5.; Wikipedia



Molecular Weight (MW)

398.29 
Formula

C18H24BrNO4 
CAS No.

155-41-9 
Storage

-20℃ for 3 years in powder form
-80℃ for 2 years in solvent
Solubility (In vitro)

DMSO: 79 mg/mL (198.3 mM) 
Water: 67 mg/mL (168.2 mM)
Ethanol: <1 mg/mL
Solubility (In vivo)

 
Synonyms

 

other peoduct :References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/19390656

In Vitro

In vitro activity


Kinase Assay:


Cell Assay

In Vivo  
Animal model  
Formulation & Dosage  
References  

TAK-242

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Author: Sodium channel

Share this post on:

product name Methscopolamine


Description: Methscopolamine is a muscarinic acetylcholine receptor blocker. Methscopolamine, a methylated derivative of scopolamine, is a muscarinic antagonist structurally similar to the neurotransmitter acetylcholine. Its mechanism of action involves blocking the muscarinic acetylcholine receptors. Methscopolamine is also commonly used as a drying agent, to dry up post-nasal drip, in cold, irritable bowel syndrome and allergy medications.

References: J Pharm Pharmacol. 1964 Oct;16:690-5.; Wikipedia



Molecular Weight (MW)

398.29 
Formula

C18H24BrNO4 
CAS No.

155-41-9 
Storage

-20℃ for 3 years in powder form
-80℃ for 2 years in solvent
Solubility (In vitro)

DMSO: 79 mg/mL (198.3 mM) 
Water: 67 mg/mL (168.2 mM)
Ethanol: <1 mg/mL
Solubility (In vivo)

 
Synonyms

 

other peoduct :References PubMed ID::http://www.ncbi.nlm.nih.gov/pubmed/19390656

In Vitro

In vitro activity


Kinase Assay:


Cell Assay

In Vivo  
Animal model  
Formulation & Dosage  
References  

TAK-242

Share this post on:

Author: Sodium channel