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product name Etizolam


Description: Etizolam is a benzodiazepine analog and a specific platelet-activating factor (PAF) antagonist with anti-anxiety activity. Etizolam is marketed under the brand name Etilaam, Etizola, Sedekopan, Etizest, Pasaden or Depas. The etizolam molecule differs from a benzodiazepine in that the benzene ring has been replaced by a thiophene ring and triazole ring has been fused, making the drug a thienotriazolodiazepine. It possesses amnesic, anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties.

References: Biol Pharm Bull. 2005 Sep;28(9):1711-6; Curr Drug Metab. 2008 Oct;9(8):827-44.



Molecular Weight (MW)

342.85 
Formula

C17H15ClN4
CAS No.

40054-69-1 
Storage

-20℃ for 3 years in powder form
-80℃ for 2 years in solvent
Solubility (In vitro)

DMSO: 26 mg/mL (75.8 mM)
Water: <1 mg/mL
Ethanol: 62 mg/mL (180.8 mM)
Solubility (In vivo)

 
Synonyms

 

other peoduct :

In Vitro

In vitro activity


Kinase Assay:


Cell Assay

In Vivo  
Animal model  
Formulation & Dosage  
References  

TIC12

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Author: Sodium channel